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Mocravimod hydrochloride
CAS No. 509088-69-1
Mocravimod hydrochloride ( KRP-203 )
产品货号. M26300 CAS No. 509088-69-1
Mocravimod Hydrochloride 是一种有效的口服活性鞘氨醇 1-磷酸受体 1 型 (S1PR1) 激动剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2001 | 有现货 |
|
| 10MG | ￥3216 | 有现货 |
|
| 25MG | ￥5370 | 有现货 |
|
| 50MG | ￥7655 | 有现货 |
|
| 100MG | ￥10368 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Mocravimod hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Mocravimod Hydrochloride 是一种有效的口服活性鞘氨醇 1-磷酸受体 1 型 (S1PR1) 激动剂。
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产品描述Mocravimod hydrochloride is an effecitive and orally active agonist of sphingosine 1-phosphate receptor type 1(S1PR1). (In Vivo):In mHC-disparate rat heart allografts, Mocravimod hydrochloride(orally; 0.1 and 1 mg/kg/day; for 100 days) prolongs graft survival and attenuates chronic rejection. Mocravimod hydrochloride ameliorates atherosclerosis in LDL-R(-/-) Mice.
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体外实验——
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体内实验Animal Model:Inbred male DA (MHC haplotype: RT1a) rats Dosage:0.1 and 1 mg/kg Administration:Orally; daily; for 100 days.Result:Prolonged graft survival and attenuated chronic rejection in mHC-disparate rat heart allografts.
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同义词KRP-203
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通路Others
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靶点Other Targets
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受体gluconeogenesis
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研究领域——
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适应症——
化学信息
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CAS Number509088-69-1
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分子量480.44
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分子式C24H27Cl2NO3S
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO : 200 mg/mL (416.28 mM)
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SMILESCl.NC(CO)(CO)CCc1ccc(Sc2cccc(OCc3ccccc3)c2)cc1Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Murray AF, et, al. Phenylpropanoid Glycerol Glucosides Attenuate Glucose Production in Hepatocytes. ACS Omega. 2019 Jun 19;4(6):10670-10676.
产品手册
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